Suche
Innovative zinc-binding inhibitors of Legionella pneumophila ProA reduce collagen and flagellin degradation, TLR5 evasion, and human lung tissue inflammation
Publikation
Scheithauer L,
Ornago C,
Selmar J,
Schütz C,
Bianchi G,
Kiefer A,
Haupenthal J,
Dellmann A,
Huynh D,
Zhang R,
Blankenfeldt W,
Hirsch A,
Steinert M
(2025)
European journal of medicinal chemistry, 296, 10.1016/j.ejmech.2025.117832, 40479898
European journal of medicinal chemistry, 296, 10.1016/j.ejmech.2025.117832, 40479898
Engineering an Artificial Myxopyronin Derivative with Enhanced Metabolic Stability via Mutasynthesis
Publikation
Kiefer A,
Voltz A,
Scherzer D,
Reberšek R,
Kany A,
Prosser G,
Neuber M,
Reiling N,
Hirsch A,
Müller R
(2025)
, 10.26434/chemrxiv-2025-q4h0n
, 10.26434/chemrxiv-2025-q4h0n
Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity
Publikation
Ropponen H,
Bader C,
Diamanti E,
Illarionov B,
Rottmann M,
Fischer M,
Witschel M,
Müller R,
Hirsch A
(2021)
ChemMedChem, 16, 13, 2089-2093, 10.1002/cmdc.202100067, 33844432
ChemMedChem, 16, 13, 2089-2093, 10.1002/cmdc.202100067, 33844432
Dipeptidic Phosphonates: Potent Inhibitors of Pseudomonas aeruginosa Elastase B Showing Efficacy in a Murine Keratitis Model
Publikation
Kiefer A,
Schütz C,
Englisch C,
Kolling D,
Speicher S,
Kany A,
Shafiei R,
Wadood N,
Aljohmani A,
Wirschem N,
Jumde R,
Klein A,
Sikandar A,
Park Y,
Krasteva-Christ G,
Yildiz D,
Abdelsamie A,
Rox K,
Köhnke J,
Müller R,
Bischoff M,
Haupenthal J,
Hirsch A
(2025)
Adv. Sci., 10.1002/advs.202411807, 39973061
Adv. Sci., 10.1002/advs.202411807, 39973061
Synthesis of New Cyclomarin Derivatives and Their Biological Evaluation towards Mycobacterium Tuberculosis and Plasmodium Falciparum
Publikation
Kiefer A,
Bader C,
Held J,
Esser A,
Rybniker J,
Empting M,
Müller R,
Kazmaier U
(2019)
Chem. Eur. J., 25, 37, 8894-8902, 10.1002/chem.201901640, 31012978
Chem. Eur. J., 25, 37, 8894-8902, 10.1002/chem.201901640, 31012978