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N -Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases
Publikation
Konstantinovic J,
Yahiaoui S,
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Kany A,
Müller R,
Koehnke J,
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J. Med. Chem., 63, 15, 8359-8368, 10.1021/acs.jmedchem.0c00584
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Discovery of the first small-molecule CsrA-RNA interaction inhibitors using biophysical screening technologies
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Maurer C,
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Avrutina O,
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Future medicinal chemistry, 8, 9, 931-47, 10.4155/fmc-2016-0033, 27253623
Future medicinal chemistry, 8, 9, 931-47, 10.4155/fmc-2016-0033, 27253623
Discovery of a novel, selective CK2 inhibitor class with an unusual basic scaffold
Publikation
Khalifa H,
ElHady A,
Liu T,
Elgaher W,
Filhol-Cochet O,
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Abadi A,
Hamed M,
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European journal of medicinal chemistry, 282, 10.1016/j.ejmech.2024.117048, 39566243
European journal of medicinal chemistry, 282, 10.1016/j.ejmech.2024.117048, 39566243
Author Correction: Octyl itaconate enhances VSVΔ51 oncolytic virotherapy by multitarget inhibition of antiviral and inflammatory pathways
Publikation
Kurmasheva N,
Said A,
Wong B,
Kinderman P,
Han X,
Rahimic A,
Kress A,
Carter-Timofte M,
Holm E,
van der Horst D,
Kollmann C,
Liu Z,
Wang C,
Hoang H,
Kovalenko E,
Chrysopoulou M,
Twayana K,
Ottosen R,
Svenningsen E,
Begnini F,
Kiib A,
Kromm F,
Weiss H,
Di Carlo D,
Muscolini M,
Higgins M,
van der Heijden M,
Arulanandam R,
Bardoul A,
Tong T,
Ozsvar A,
Hou W,
Schack V,
Holm C,
Zheng Y,
Ruzek M,
Kalucka J,
La Vega L,
Elgaher W,
Korshoej A,
Lin R,
Hiscott J,
Poulsen T,
O'Neill L,
Roy D,
Rinschen M,
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Diallo J,
Farin H,
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Nat Commun, 15, 1, 10.1038/s41467-024-55044-w, 39702301
Nat Commun, 15, 1, 10.1038/s41467-024-55044-w, 39702301
Novel and Extremely Sensitive NiAl2O4-NiO Nanostructures on an ITO Sensing Electrode for Enhanced Detection of Ascorbic Acid
Publikation
Hammami A,
Bardaoui A,
Eissa S,
Elgaher W,
Chtourou R,
Messaoud O
(2024)
Molecules (Basel, Switzerland), 29, 12, 10.3390/molecules29122837, 38930902
Molecules (Basel, Switzerland), 29, 12, 10.3390/molecules29122837, 38930902
Octyl itaconate enhances VSVΔ51 oncolytic virotherapy by multitarget inhibition of antiviral and inflammatory pathways
Publikation
Kurmasheva N,
Said A,
Wong B,
Kinderman P,
Han X,
Rahimic A,
Kress A,
Carter-Timofte M,
Holm E,
van der Horst D,
Kollmann C,
Liu Z,
Wang C,
Hoang H,
Kovalenko E,
Chrysopoulou M,
Twayana K,
Ottosen R,
Svenningsen E,
Begnini F,
Kiib A,
Kromm F,
Weiss H,
Di Carlo D,
Muscolini M,
Higgins M,
van der Heijden M,
Arulanandam R,
Bardoul A,
Tong T,
Ozsvar A,
Hou W,
Schack V,
Holm C,
Zheng Y,
Ruzek M,
Kalucka J,
La Vega L,
Elgaher W,
Korshoej A,
Lin R,
Hiscott J,
Poulsen T,
O'Neill L,
Roy D,
Rinschen M,
van Montfoort N,
Diallo J,
Farin H,
Alain T,
Olagnier D
(2024)
Nat Commun, 15, 1, 10.1038/s41467-024-48422-x, 38750019
Nat Commun, 15, 1, 10.1038/s41467-024-48422-x, 38750019
Citraconic acid and derivatives thereof for use as a medicament
Publikation
Frank Pessler,
Fangfang Chen,
Moritz Winterhoff,
Konrad Büssow,
Wulf Blankenfeldt,
Anna Hirsch,
Walid A. M. Elgaher
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Patent, A61K31/122; A61K31/194; A61P31/16; C07C57/42; C07C61/20; C07C69/593;, US20240368065A1
Patent, A61K31/122; A61K31/194; A61P31/16; C07C57/42; C07C61/20; C07C69/593;, US20240368065A1
3D bioprinting ofE. coliMG1655 biofilms on human lung epithelial cells for building complexin vitroinfection models
Publikation
Aliyazdi S,
Frisch S,
Hidalgo A,
Frank N,
Krug D,
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Vogt T,
Loretz B,
Lehr C
(2023)
Biofabrication, 15, 3, 10.1088/1758-5090/acd95e, 37236174
Biofabrication, 15, 3, 10.1088/1758-5090/acd95e, 37236174
Korrektur der absoluten Konfiguration von Chelocardin und Amidochelocardin
Publikation
Sikandar A,
Popoff A,
Jumde R,
Mándi A,
Kaur A,
Elgaher W,
Rosenberger L,
Hüttel S,
Jansen R,
Hunter M,
Köhnke J,
Hirsch A,
Kurtán T,
Müller R
(2023)
Angewandte Chemie (Weinheim an der Bergstrasse, Germany), 135, 40, 10.1002/ange.202306437
Angewandte Chemie (Weinheim an der Bergstrasse, Germany), 135, 40, 10.1002/ange.202306437
Crystobactamides
Publikation
Sascha Baumann,
Jennifer Herrmann,
Kathrin Mohr,
Heinrich Steinmetz,
Klaus Gerth,
Ritesh Raju,
Rolf Müller,
Rolf W. Hartmann,
Mostafa Hamed,
Walid A. M. Elgaher,
Maria Moreno,
Franziska Gille,
Liang Liang Wang,
Andreas Kirschning,
Stephan Huettel
(2022)
Patent, C07C237/42; C07C237/44; C07K5/065; C07K7/06; C12N15/52; C12P13/02; A61K38/00, US11225503B2
Patent, C07C237/42; C07C237/44; C07K5/065; C07K7/06; C12N15/52; C12P13/02; A61K38/00, US11225503B2