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Targeting the Plasmodium falciparum IspE Enzyme
Publikation
Diamanti E,
Steinbach A,
Carvalho L,
Ropponen H,
Lacour A,
Hamid R,
Eisa S,
Bravo P,
Bousis S,
Illarionov B,
Fischer M,
Hamed M,
Bach N,
Rottmann M,
Held J,
Witschel M,
Sieber S,
Hirsch A
(2024)
ACS omega, 9, 44, 44465-44473, 10.1021/acsomega.4c06038, 39524657
ACS omega, 9, 44, 44465-44473, 10.1021/acsomega.4c06038, 39524657
Behavioral and electrophysiological responses of the male medfly, Ceratitis capitata, to thymol and carvacrol ethers
Publikation
Tabanca N,
Cloonan K,
Nesterkina M,
Gill M,
Montgomery W,
Kravchenko I,
Kendra P
(2024)
Pest management science, 10.1002/ps.8324, 39096116
Pest management science, 10.1002/ps.8324, 39096116
Evaluation of ketoclomazone and its analogues as inhibitors of 1-deoxy-d-xylulose 5-phosphate synthases and other thiamine diphosphate (ThDP)-dependent enzymes
Publikation
Chan A,
Ho T,
Fathoni I,
Hamid R,
Hirsch A,
Saliba K,
Leeper F
(2024)
RSC Med. Chem., 15, 5, 1773-1781, 10.1039/D4MD00083H, 38784473
RSC Med. Chem., 15, 5, 1773-1781, 10.1039/D4MD00083H, 38784473
Studying Target-Engagement of Anti-Infectives by Solvent-Induced Protein Precipitation and Quantitative Mass Spectrometry
Publikation
Bizzarri L,
Steinbrunn D,
Quennesson T,
Lacour A,
Bianchino G,
Bravo P,
Chaignon P,
Lohse J,
Mäser P,
Seemann M,
van Calenbergh S,
Hirsch A,
Hahne H
(2024)
ACS Infect. Dis., 10, 12, 4087-4102, 10.1021/acsinfecdis.4c00417, 39566904
ACS Infect. Dis., 10, 12, 4087-4102, 10.1021/acsinfecdis.4c00417, 39566904
Synthesis and Structure of a Coordination Polymer of Ni(II) with 2-(4-Bromophenoxy)acetohydrazide
Publikation
Martsynko ?,
Nesterkina M,
Finik ?,
Tsymbaliuk K,
Dyakonenko V,
Shishkina S,
Kravchenko I
(2024)
Molbank, 2024, 2, 10.3390/M1819
Molbank, 2024, 2, 10.3390/M1819
Towards the evaluation in an animal disease model: Fluorinated 17β-HSD1 inhibitors showing strong activity towards both the human and the rat enzyme
Publikation
Abdelsamie A,
Bey E,
Gargano E,
van Koppen C,
Empting M,
Frotscher M
(2015)
European journal of medicinal chemistry, 103, 56-68, 10.1016/j.ejmech.2015.08.030, 26322835
European journal of medicinal chemistry, 103, 56-68, 10.1016/j.ejmech.2015.08.030, 26322835
Novel PqsR Inverse Agonists
Publikation
Hamed M
(2015)
Patent, EP 201523196
Patent, EP 201523196
Fragment growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin
Publikation
Mondal M,
Groothuis D,
Hirsch A
(2015)
, 10.1039/C5MD00157A
, 10.1039/C5MD00157A
Validation of a homology model of Mycobacterium tuberculosis DXS: rationalization of observed activities of thiamine derivatives as potent inhibitors of two orthologues of DXS
Publikation
Masini T,
Lacy B,
Monjas L,
Hawksley D,
Voogd A,
Illarionov B,
Iqbal A,
Leeper F,
Fischer M,
Kontoyianni M,
Hirsch A
(2015)
Organic & biomolecular chemistry, 13, 46, 11263-77, 10.1039/c5ob01666e, 26411373
Organic & biomolecular chemistry, 13, 46, 11263-77, 10.1039/c5ob01666e, 26411373
Structure-based design of potent small-molecule binders to the S-component of the ECF transporter for thiamine
Publikation
Swier L,
Monjas L,
Guskov A,
Voogd A,
Erkens G,
slotboom d,
Hirsch A
(2015)
ChemBioChem, 16, 5, 819-26, 10.1002/cbic.201402673, 25676607
ChemBioChem, 16, 5, 819-26, 10.1002/cbic.201402673, 25676607