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Publikation
Aleksandrova A,
Nesterkina M,
Gvozdii S,
Kravchenko I
(2020)
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules that Target Bacterial Glucosyltransferase
Publikation
Hartman A,
Jumde V,
Elgaher W,
Te Poele E,
Dijkhuizen L,
Hirsch A
(2020)
ChemMedChem, 10.1002/cmdc.202000222, 32542998
ChemMedChem, 10.1002/cmdc.202000222, 32542998
Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination
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Vlag R,
Yagiz Unver M,
Felicetti T,
Twarda-Clapa A,
Kassim F,
Ermis C,
Neochoritis C,
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Dömling A,
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Hirsch A
(2020)
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
2-Propyl-N′-[1,7,7-trimethylbicyclo[2.2.1]hept-2-ylidene]pentanehydrazide
Publikation
Nesterkina M,
Barbalat D,
Rakipov I,
Kravchenko I
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Molbank, 2020, 4, 10.3390/M1164
Molbank, 2020, 4, 10.3390/M1164
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction
Publikation
Federica Mancini,
M. Yagiz Unver,
Walid A. M. Elgaher,
Varsha R. Jumde,
Alaa Alhayek,
Peer Lukat,
Jennifer Herrmann,
Martin D. Witte,
Matthias Köck,
Wulf Blankenfeldt,
Rolf Müller,
Hirsch A
(2020)
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Design, synthesis and pharmacological profile of (−)-verbenone hydrazones
Publikation
Nesterkina M,
Barbalat D,
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Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
7-Hydroxycoumarins are Affinity-based Fluorescent Probes for Competitive Binding Studies of Macrophage Migration Inhibitory Factor
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Xiao Z,
Chen D,
Song S,
van der Vlag R,
van der Wouden P,
van Merkerk R,
Cool R,
Hirsch A,
Melgert B,
Quax W,
Poelarends G,
Dekker F
(2020)
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Restriction-Free Construction of a Phage-Presented Very Short Macrocyclic Peptide Library
Publikation
Jakob V,
Helmsing S,
Hust M,
Empting M
(2020)
Methods in molecular biology (Clifton, N.J.), 2070, 95-113, 10.1007/978-1-4939-9853-1_6, 31625092
Methods in molecular biology (Clifton, N.J.), 2070, 95-113, 10.1007/978-1-4939-9853-1_6, 31625092
Semisynthesis and biological evaluation of amidochelocardin derivatives as broad-spectrum antibiotics
Publikation
Grandclaudon C,
Birudukota N,
Elgaher W,
Jumde R,
Yahiaoui S,
Arisetti N,
Hennessen F,
Hüttel S,
Stadler M,
Herrmann J,
Miethke M,
Hartmann R,
Müller R,
Hirsch A,
Brönstrup M
(2020)
European journal of medicinal chemistry, 188, 10.1016/j.ejmech.2019.112005, 31911294
European journal of medicinal chemistry, 188, 10.1016/j.ejmech.2019.112005, 31911294
Novel PqsR Inverse Agonists
Publikation
Hamed M,
Ahmed S,
Empting. M.,
Schütz C,
Hartmann R,
Röhrig T,
Kany A,
Hirsch A
(2020)
Patent, EP20150119
Patent, EP20150119