![[Translate to Deutsch:]](/fileadmin/HIPS/__processed__/3/9/csm_HIPS_50243_47cfe3711c.jpg "[Translate to Deutsch:]")
Suche
Rational Adaptation of L3MBTL1 Inhibitors to Create Small-Molecule Cbx7 Antagonists
Publikation
Simhadri C,
Daze K,
Douglas S,
Milosevich N,
Monjas L,
Dev A,
Brown T,
Hirsch A,
Wulff J,
Hof F
(2019)
ChemMedChem, 14, 15, 1444-1456, 10.1002/cmdc.201900021, 31254321
ChemMedChem, 14, 15, 1444-1456, 10.1002/cmdc.201900021, 31254321
Fragment-Based Discovery of a Qualified Hit Targeting the Latency-Associated Nuclear Antigen of the Oncogenic Kaposi's Sarcoma-Associated Herpesvirus/Human Herpesvirus 8
Publikation
Kirsch P,
Jakob V,
Oberhausen K,
Stein S,
Cucarro I,
Schulz T,
Empting M
(2019)
Journal of medicinal chemistry, 62, 8, 3924-3939, 10.1021/acs.jmedchem.8b01827, 30888817
Journal of medicinal chemistry, 62, 8, 3924-3939, 10.1021/acs.jmedchem.8b01827, 30888817
Protein-Templated Dynamic Combinatorial Chemistry: Brief Overview and Experimental Protocol
Publikation
Hartman A,
Gierse R,
Hirsch A
(2019)
European journal of organic chemistry, 2019, 22, 3581-3590, 10.1002/ejoc.201900327, 31680778
European journal of organic chemistry, 2019, 22, 3581-3590, 10.1002/ejoc.201900327, 31680778
Replacement of an Indole Scaffold Targeting Human 15-Lipoxygenase-1 Using Combinatorial Chemistry
Publikation
Prismawan D,
van der Vlag R,
Guo H,
Dekker F,
Hirsch A
(2019)
HCA, 102, 5, 10.1002/hlca.201900040, 31231138
HCA, 102, 5, 10.1002/hlca.201900040, 31231138
Spray-drying of inhalable, multifunctional formulations for the treatment of biofilms formed in cystic fibrosis
Publikation
Lababidi N,
Ofosu Kissi E,
Elgaher W,
Sigal V,
Haupenthal J,
Schwarz B,
Hirsch A,
Rades T,
Schneider M
(2019)
Journal of Controlled Release, 314, 62-71, 10.1016/j.jconrel.2019.10.038
Journal of Controlled Release, 314, 62-71, 10.1016/j.jconrel.2019.10.038
Studying Target-Engagement of Anti-Infectives by Solvent-Induced Protein Precipitation and Quantitative Mass Spectrometry
Publikation
Bizzarri L,
Steinbrunn D,
Quennesson T,
Lacour A,
Bianchino G,
Bravo P,
Chaignon P,
Lohse J,
Mäser P,
Seemann M,
van Calenbergh S,
Hirsch A,
Hahne H
(2024)
ACS Infect. Dis., 10, 12, 4087-4102, 10.1021/acsinfecdis.4c00417, 39566904
ACS Infect. Dis., 10, 12, 4087-4102, 10.1021/acsinfecdis.4c00417, 39566904
Synthesis and Structure of a Coordination Polymer of Ni(II) with 2-(4-Bromophenoxy)acetohydrazide
Publikation
Martsynko ?,
Nesterkina M,
Finik ?,
Tsymbaliuk K,
Dyakonenko V,
Shishkina S,
Kravchenko I
(2024)
Molbank, 2024, 2, 10.3390/M1819
Molbank, 2024, 2, 10.3390/M1819
Target repurposing unravels avermectins and derivatives as novel antibiotics inhibiting energy-coupling factor transporters (ECFTs)
Publikation
Haupenthal J,
Rafehi M,
Kany A,
Lespine A,
Stefan K,
Hirsch* A,
Stefan* S
(2024)
Arch. Pharm., 10.1002/ardp.202400267, 38896404
Arch. Pharm., 10.1002/ardp.202400267, 38896404
Not Every Hit-Identification Technique Works on 1-Deoxy-d-Xylulose 5-Phosphate Synthase (DXPS): Making the Most of a Virtual Screening Campaign
Publikation
Johannsen S,
Gierse R,
Olshanova A,
Smerznak E,
Laggner C,
Eschweiler L,
Adeli Z,
Hamid R,
Alhayek A,
Reiling N,
Haupenthal J,
Hirsch A
(2023)
ChemMedChem, 10.1002/cmdc.202200590, 36896721
ChemMedChem, 10.1002/cmdc.202200590, 36896721
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
Publikation
Ropponen H,
Diamanti E,
Johannsen S,
Illarionov B,
Hamid R,
Jaki M,
Sass P,
Fischer M,
Haupenthal J,
Hirsch A
(2023)
ChemMedChem, 10.1002/cmdc.202300346, 37718320
ChemMedChem, 10.1002/cmdc.202300346, 37718320