Suche
9,10-Anthraquinone Dithiocarbamates as Potential Pharmaceutical Substances with Pleiotropic Actions: Computerized Prediction of Biological Activity and Experimental Validation
Publikation
Stasevich M,
Zvarich V,
Novikov V,
Zagorodnyaya S,
Povnitsa O,
Chaika M,
Nesterkina M,
Kravchenko I,
Druzhilovskii D,
Poroikov V
(2020)
Pharm Chem J, 53, 10, 905-913, 10.1007/s11094-020-02098-x
Pharm Chem J, 53, 10, 905-913, 10.1007/s11094-020-02098-x
Phytochemical analysis and anti-inflammatory activity of Cladophora aegagropila extract
Publikation
Aleksandrova A,
Nesterkina M,
Gvozdii S,
Kravchenko I
(2020)
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules that Target Bacterial Glucosyltransferase
Publikation
Hartman A,
Jumde V,
Elgaher W,
Te Poele E,
Dijkhuizen L,
Hirsch A
(2020)
ChemMedChem, 10.1002/cmdc.202000222, 32542998
ChemMedChem, 10.1002/cmdc.202000222, 32542998
Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination
Publikation
Vlag R,
Yagiz Unver M,
Felicetti T,
Twarda-Clapa A,
Kassim F,
Ermis C,
Neochoritis C,
Musielak B,
Labuzek B,
Dömling A,
Holak T,
Hirsch A
(2020)
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
2-Propyl-N′-[1,7,7-trimethylbicyclo[2.2.1]hept-2-ylidene]pentanehydrazide
Publikation
Nesterkina M,
Barbalat D,
Rakipov I,
Kravchenko I
(2020)
Molbank, 2020, 4, 10.3390/M1164
Molbank, 2020, 4, 10.3390/M1164
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction
Publikation
Federica Mancini,
M. Yagiz Unver,
Walid A. M. Elgaher,
Varsha R. Jumde,
Alaa Alhayek,
Peer Lukat,
Jennifer Herrmann,
Martin D. Witte,
Matthias Köck,
Wulf Blankenfeldt,
Rolf Müller,
Hirsch A
(2020)
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Design, synthesis and pharmacological profile of (−)-verbenone hydrazones
Publikation
Nesterkina M,
Barbalat D,
Kravchenko I
(2020)
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
7-Hydroxycoumarins are Affinity-based Fluorescent Probes for Competitive Binding Studies of Macrophage Migration Inhibitory Factor
Publikation
Xiao Z,
Chen D,
Song S,
van der Vlag R,
van der Wouden P,
van Merkerk R,
Cool R,
Hirsch A,
Melgert B,
Quax W,
Poelarends G,
Dekker F
(2020)
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
Publikation
Ropponen H,
Diamanti E,
Johannsen S,
Illarionov B,
Hamid R,
Jaki M,
Sass P,
Fischer M,
Haupenthal J,
Hirsch A
(2023)
ChemMedChem, 10.1002/cmdc.202300346, 37718320
ChemMedChem, 10.1002/cmdc.202300346, 37718320
Genotoxic and mutational potential of monocyclic terpenoids (carvacrol, carvone and thymol) in Drosophila melanogaster
Publikation
Nesterkina M,
Bilokon S,
Alieksieieva T,
Kravchenko I,
Hirsch A
(2023)
Toxicol. Rep., 10, 10.1016/j.toxrep.2023.02.009
Toxicol. Rep., 10, 10.1016/j.toxrep.2023.02.009