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Researchers in HIPS Laboratory

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Searched for "drug". Displaying results 701 to 710 of 812.

BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application

Publication
Della Volpe S, Listro R, Parafioriti M, Di Giacomo M, Rossi D, Ambrosio F, Costa G, Alcaro S, Ortuso F, Hirsch A, Vasile F, Collina S (2020)
ACS medicinal chemistry letters, 11, 5, 883-888, 10.1021/acsmedchemlett.9b00659, 32435400

Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach

Publication
Konstantinidou M, Magari F, Sutanto F, Haupenthal J, Jumde R, Ünver M, Heine A, Camacho C, Hirsch A, Klebe G, Dömling A (2020)
ChemMedChem, 15, 8, 680-684, 10.1002/cmdc.202000024

Evaluation of Bacterial RNA Polymerase Inhibitors in a Staphylococcus aureus-Based Wound Infection Model in SKH1 Mice

Publication
Haupenthal J, Kautz Y, Elgaher W, Pätzold L, Röhrig T, Laschke M, Tschernig T, Hirsch A, Molodtsov V, Murakami K, Hartmann R, Bischoff M (2020)
ACS infectious diseases, 6, 10, 2573-2581, 10.1021/acsinfecdis.0c00034, 32886885

Flotillin-mediated membrane fluidity controls peptidoglycan synthesis and MreB movement

Publication
Zielinska A, Savietto A, Sousa Borges A, Martinez D, Berbon M, Roelofsen J, Hartman A, Boer R, van der Klei I, Hirsch A, Habenstein B, Bramkamp M, Scheffers D (2020)
eLife, 9, 10.7554/eLife.57179

Synthesis and Evaluation on Anticonvulsant and Antidepressant Activities of Naphthoquinone Derivatives Containing Pyrazole and Pyrimidine Fragments

Publication
Polish N, Nesterkina M, Marintsova N, Karkhut A, Kravchenko I, Novikov V, Khairulin A (2020)
ACSi, 67, 3, 934-939, 10.17344/acsi.2020.5938

Tracheal brush cells release acetylcholine in response to bitter tastants for paracrine and autocrine signaling

Publication
Hollenhorst M, Jurastow I, Nandigama R, Appenzeller S, Li L, Vogel J, Wiederhold S, Althaus M, Empting M, Altmüller J, Hirsch A, Flockerzi V, Canning B, Saliba A, Krasteva-Christ G (2020)
FASEB j., 34, 1, 316-332, 10.1096/fj.201901314RR

(2S,5R)-2-Isopropyl-5-methylcyclohexanone Hydrazones

Publication
Nesterkina M, Barbalat D, Zheltvay I, Rakipov I, Atakay M, Salih B, Kravchenko I (2019)
Molbank, 2019, 2, 10.3390/M1062

Anti-inflammatory and analgesic activity of ointment based on dense ginger extract (Zingiber officinale)

Publication
Kravchenko I, Eberle L, Nesterkina M, Kobernik A (2019)
J Herbmed Pharmacol, 8, 2, 126-132, 10.15171/jhp.2019.20

Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof-of-Principle

Publication
Hamed M, Abdelsamie A, Rox K, Schütz C, Kany A, Röhrig T, Schmelz S, Blankenfeldt W, Arce-Rodriguez A, Borrero-de Acuña J, Jahn D, Rademacher J, Ringshausen F, Cramer N, Tümmler B, Hirsch A, Hartmann R, Empting M (2023)
Adv. Sci., Online, 10.1002/advs.202204443

Design of thiamine analogues for inhibition of thiamine diphosphate (ThDP)-dependent enzymes: Systematic investigation through Scaffold-Hopping and C2-Functionalisation

Publication
Chan A, Ho T, Irfan R, Hamid R, Rudge E, Iqbal A, Turner A, Hirsch A., Leeper F (2023)
Bioorganic chemistry, 138, 10.1016/j.bioorg.2023.106602