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Researchers in HIPS Laboratory

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Searched for "drug". Displaying results 651 to 660 of 750.

Design and synthesis of thiamine analogues to study their binding to the ECF transporter for thiamine in bacteria

Publication
Monjas L, Swier L, Voogd A, Oudshoorn R, Hirsch A, Slotboom D (2016)
Med. Chem. Commun., 7, 5, 966-971, 10.1039/C6MD00022C

Dissecting the Multiple Roles of PqsE in Pseudomonas aeruginosa Virulence by Discovery of Small Tool Compounds

Publication
Zender M, Witzgall F, Drees S, Weidel E, Maurer C, Fetzner S, Blankenfeldt W, Empting M, Hartmann R (2016)
ACS chemical biology, 10.1021/acschembio.6b00156, 27082157

Discovery and Structure-Based Optimization of 2-Ureidothiophene-3-carboxylic Acids as Dual Bacterial RNA Polymerase and Viral Reverse Transcriptase Inhibitors

Publication
Elgaher W, Sharma K, Haupenthal J, Saladini F, Pires M, Real E, Mely Y, Hartmann R (2016)
Journal of medicinal chemistry, 10.1021/acs.jmedchem.6b00730, 27339173

Structure-Activity Relationships of 2-Sufonylpyrimidines as Quorum-Sensing Inhibitors to Tackle Biofilm Formation and eDNA Release of Pseudomonas aeruginosa

Publication
Thomann A, Brengel C, Börger C, Kail D, Steinbach A, Empting M, Hartmann R (2016)
ChemMedChem, 11, 22, 2522-2533, 10.1002/cmdc.201600419, 27731921

Furoates and thenoates inhibit pyruvate dehydrogenase kinase 2 allosterically by binding to its pyruvate regulatory site

Publication
Masini T, Birkaya B, van Dijk S, Mondal M, Hekelaar J, Jäger M, van Terwisscha Scheltinga A, Patel M, Hirsch A, Moman E (2016)
Journal of enzyme inhibition and medicinal chemistry, 31, sup4, 170-175, 10.1080/14756366.2016.1201812, 27435185

Synthesis and Anticonvulsant Activity of Menthyl γ-Aminobutyrate

Publication
Nesterkina M, Kravchenko I (2016)
Chem Nat Compd, 52, 2, 237-239, 10.1007/s10600-016-1604-9

Synthesis and Pharmacological Properties of Novel Esters Based on Monocyclic Terpenes and GABA

Publication
Nesterkina M, Kravchenko I (2016)
Pharmaceuticals (Basel, Switzerland), 9, 2, 10.3390/ph9020032, 27304960

Analgesic Activity of Novel GABA Esters after Transdermal Delivery

Publication
Nesterkina M, Kravchenko I (2016)
Nat. Prod. Commun., 11, 10, 10.1177/1934578X1601101001

Single-domain antibodies for biomedical applications

Publication
Krah S, Schröter C, Zielonka S, Empting M, Valldorf B, Kolmar H (2016)
Immunopharmacol. Immunotoxicol., 38, 1, 21-8, 10.3109/08923973.2015.1102934, 26551147

Synthesis and Anticonvulsant Activity of New Calix[4]Arene Derivatives Containing Gamma-Aminobutyric Acid Moieties

Publication
Nesterkina M, Alekseeva E, Kravchenko I (2016)
Pharm Chem J, 49, 12, 825-829, 10.1007/s11094-016-1380-7