Search
Discovery of Novel Latency-Associated Nuclear Antigen Inhibitors as Antiviral Agents Against Kaposi's Sarcoma-Associated Herpesvirus
Publication
Kirsch P,
Jakob V,
Elgaher W,
Walt C,
Oberhausen K,
Schulz T,
Empting M
(2020)
ACS chemical biology, 15, 2, 388-395, 10.1021/acschembio.9b00845, 31944659
ACS chemical biology, 15, 2, 388-395, 10.1021/acschembio.9b00845, 31944659
Discovery of Small-Molecule Stabilizers of 14-3-3 Protein-Protein Interactions via Dynamic Combinatorial Chemistry
Publication
Hartman A,
Elgaher W,
Hertrich N,
Andrei S,
Ottmann C,
Hirsch A
(2020)
ACS medicinal chemistry letters, 11, 5, 1041-1046, 10.1021/acsmedchemlett.9b00541, 32435423
ACS medicinal chemistry letters, 11, 5, 1041-1046, 10.1021/acsmedchemlett.9b00541, 32435423
QSAR models for analgesic activity prediction of terpenes and their derivatives
Publication
Nesterkina M,
Ognichenko L,
Shyrykalova A,
Kravchenko I,
Kuz’min V
(2020)
Struct Chem, 31, 3, 947-954, 10.1007/s11224-019-01479-7
Struct Chem, 31, 3, 947-954, 10.1007/s11224-019-01479-7
9,10-Anthraquinone Dithiocarbamates as Potential Pharmaceutical Substances with Pleiotropic Actions: Computerized Prediction of Biological Activity and Experimental Validation
Publication
Stasevich M,
Zvarich V,
Novikov V,
Zagorodnyaya S,
Povnitsa O,
Chaika M,
Nesterkina M,
Kravchenko I,
Druzhilovskii D,
Poroikov V
(2020)
Pharm Chem J, 53, 10, 905-913, 10.1007/s11094-020-02098-x
Pharm Chem J, 53, 10, 905-913, 10.1007/s11094-020-02098-x
Phytochemical analysis and anti-inflammatory activity of Cladophora aegagropila extract
Publication
Aleksandrova A,
Nesterkina M,
Gvozdii S,
Kravchenko I
(2020)
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
J Herbmed Pharmacol, 9, 1, 81-85, 10.15171/jhp.2020.12
Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules that Target Bacterial Glucosyltransferase
Publication
Hartman A,
Jumde V,
Elgaher W,
Te Poele E,
Dijkhuizen L,
Hirsch A
(2020)
ChemMedChem, 10.1002/cmdc.202000222, 32542998
ChemMedChem, 10.1002/cmdc.202000222, 32542998
Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination
Publication
Vlag R,
Yagiz Unver M,
Felicetti T,
Twarda-Clapa A,
Kassim F,
Ermis C,
Neochoritis C,
Musielak B,
Labuzek B,
Dömling A,
Holak T,
Hirsch A
(2020)
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
2-Propyl-N′-[1,7,7-trimethylbicyclo[2.2.1]hept-2-ylidene]pentanehydrazide
Publication
Nesterkina M,
Barbalat D,
Rakipov I,
Kravchenko I
(2020)
Molbank, 2020, 4, 10.3390/M1164
Molbank, 2020, 4, 10.3390/M1164
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction
Publication
Federica Mancini,
M. Yagiz Unver,
Walid A. M. Elgaher,
Varsha R. Jumde,
Alaa Alhayek,
Peer Lukat,
Jennifer Herrmann,
Martin D. Witte,
Matthias Köck,
Wulf Blankenfeldt,
Rolf Müller,
Hirsch A
(2020)
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Design, synthesis and pharmacological profile of (−)-verbenone hydrazones
Publication
Nesterkina M,
Barbalat D,
Kravchenko I
(2020)
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103