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François Diederich – In Memoriam**
Publication
Hof F,
Hirsch A
(2020)
ChemMedChem, 10.1002/cmdc.202000920
ChemMedChem, 10.1002/cmdc.202000920
BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR Application
Publication
Della Volpe S,
Listro R,
Parafioriti M,
Di Giacomo M,
Rossi D,
Ambrosio F,
Costa G,
Alcaro S,
Ortuso F,
Hirsch A,
Vasile F,
Collina S
(2020)
ACS medicinal chemistry letters, 11, 5, 883-888, 10.1021/acsmedchemlett.9b00659, 32435400
ACS medicinal chemistry letters, 11, 5, 883-888, 10.1021/acsmedchemlett.9b00659, 32435400
Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach
Publication
Konstantinidou M,
Magari F,
Sutanto F,
Haupenthal J,
Jumde R,
Ünver M,
Heine A,
Camacho C,
Hirsch A,
Klebe G,
Dömling A
(2020)
ChemMedChem, 15, 8, 680-684, 10.1002/cmdc.202000024
ChemMedChem, 15, 8, 680-684, 10.1002/cmdc.202000024
Evaluation of Bacterial RNA Polymerase Inhibitors in a Staphylococcus aureus-Based Wound Infection Model in SKH1 Mice
Publication
Haupenthal J,
Kautz Y,
Elgaher W,
Pätzold L,
Röhrig T,
Laschke M,
Tschernig T,
Hirsch A,
Molodtsov V,
Murakami K,
Hartmann R,
Bischoff M
(2020)
ACS infectious diseases, 6, 10, 2573-2581, 10.1021/acsinfecdis.0c00034, 32886885
ACS infectious diseases, 6, 10, 2573-2581, 10.1021/acsinfecdis.0c00034, 32886885
Flotillin-mediated membrane fluidity controls peptidoglycan synthesis and MreB movement
Publication
Zielinska A,
Savietto A,
Sousa Borges A,
Martinez D,
Berbon M,
Roelofsen J,
Hartman A,
Boer R,
van der Klei I,
Hirsch A,
Habenstein B,
Bramkamp M,
Scheffers D
(2020)
eLife, 9, 10.7554/eLife.57179
eLife, 9, 10.7554/eLife.57179
Synthesis and Evaluation on Anticonvulsant and Antidepressant Activities of Naphthoquinone Derivatives Containing Pyrazole and Pyrimidine Fragments
Publication
Polish N,
Nesterkina M,
Marintsova N,
Karkhut A,
Kravchenko I,
Novikov V,
Khairulin A
(2020)
ACSi, 67, 3, 934-939, 10.17344/acsi.2020.5938
ACSi, 67, 3, 934-939, 10.17344/acsi.2020.5938
Tracheal brush cells release acetylcholine in response to bitter tastants for paracrine and autocrine signaling
Publication
Hollenhorst M,
Jurastow I,
Nandigama R,
Appenzeller S,
Li L,
Vogel J,
Wiederhold S,
Althaus M,
Empting M,
Altmüller J,
Hirsch A,
Flockerzi V,
Canning B,
Saliba A,
Krasteva-Christ G
(2020)
FASEB j., 34, 1, 316-332, 10.1096/fj.201901314RR
FASEB j., 34, 1, 316-332, 10.1096/fj.201901314RR
(2S,5R)-2-Isopropyl-5-methylcyclohexanone Hydrazones
Publication
Nesterkina M,
Barbalat D,
Zheltvay I,
Rakipov I,
Atakay M,
Salih B,
Kravchenko I
(2019)
Molbank, 2019, 2, 10.3390/M1062
Molbank, 2019, 2, 10.3390/M1062
Anti-inflammatory and analgesic activity of ointment based on dense ginger extract (Zingiber officinale)
Publication
Kravchenko I,
Eberle L,
Nesterkina M,
Kobernik A
(2019)
J Herbmed Pharmacol, 8, 2, 126-132, 10.15171/jhp.2019.20
J Herbmed Pharmacol, 8, 2, 126-132, 10.15171/jhp.2019.20
Rational Adaptation of L3MBTL1 Inhibitors to Create Small-Molecule Cbx7 Antagonists
Publication
Simhadri C,
Daze K,
Douglas S,
Milosevich N,
Monjas L,
Dev A,
Brown T,
Hirsch A,
Wulff J,
Hof F
(2019)
ChemMedChem, 14, 15, 1444-1456, 10.1002/cmdc.201900021, 31254321
ChemMedChem, 14, 15, 1444-1456, 10.1002/cmdc.201900021, 31254321