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Bicyclic enol cyclocarbamates inhibit penicillin-binding proteins
Publication
Dockerty P,
Edens J,
Tol M,
Morales Angeles D,
Domenech A,
Liu Y,
Hirsch A,
Veening J,
Scheffers D,
Witte M
(2017)
Organic & biomolecular chemistry, 15, 4, 894-910, 10.1039/c6ob01664b, 28045164
Organic & biomolecular chemistry, 15, 4, 894-910, 10.1039/c6ob01664b, 28045164
Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination
Publication
Vlag R,
Yagiz Unver M,
Felicetti T,
Twarda-Clapa A,
Kassim F,
Ermis C,
Neochoritis C,
Musielak B,
Labuzek B,
Dömling A,
Holak T,
Hirsch A
(2020)
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
ChemMedChem, 15, 4, 370-375, 10.1002/cmdc.201900574
2-Propyl-N′-[1,7,7-trimethylbicyclo[2.2.1]hept-2-ylidene]pentanehydrazide
Publication
Nesterkina M,
Barbalat D,
Rakipov I,
Kravchenko I
(2020)
Molbank, 2020, 4, 10.3390/M1164
Molbank, 2020, 4, 10.3390/M1164
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction
Publication
Federica Mancini,
M. Yagiz Unver,
Walid A. M. Elgaher,
Varsha R. Jumde,
Alaa Alhayek,
Peer Lukat,
Jennifer Herrmann,
Martin D. Witte,
Matthias Köck,
Wulf Blankenfeldt,
Rolf Müller,
Hirsch A
(2020)
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Chemistry – A European Journal, 26, 64, 10.1002/chem.202086462
Design, synthesis and pharmacological profile of (−)-verbenone hydrazones
Publication
Nesterkina M,
Barbalat D,
Kravchenko I
(2020)
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
Open Chemistry, 18, 1, 943-950, 10.1515/chem-2020-0103
7-Hydroxycoumarins are Affinity-based Fluorescent Probes for Competitive Binding Studies of Macrophage Migration Inhibitory Factor
Publication
Xiao Z,
Chen D,
Song S,
van der Vlag R,
van der Wouden P,
van Merkerk R,
Cool R,
Hirsch A,
Melgert B,
Quax W,
Poelarends G,
Dekker F
(2020)
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Journal of medicinal chemistry, 10.1021/acs.jmedchem.0c01160, 32940040
Restriction-Free Construction of a Phage-Presented Very Short Macrocyclic Peptide Library
Publication
Jakob V,
Helmsing S,
Hust M,
Empting M
(2020)
Methods in molecular biology (Clifton, N.J.), 2070, 95-113, 10.1007/978-1-4939-9853-1_6, 31625092
Methods in molecular biology (Clifton, N.J.), 2070, 95-113, 10.1007/978-1-4939-9853-1_6, 31625092
Semisynthesis and biological evaluation of amidochelocardin derivatives as broad-spectrum antibiotics
Publication
Grandclaudon C,
Birudukota N,
Elgaher W,
Jumde R,
Yahiaoui S,
Arisetti N,
Hennessen F,
Hüttel S,
Stadler M,
Herrmann J,
Miethke M,
Hartmann R,
Müller R,
Hirsch A,
Brönstrup M
(2020)
European journal of medicinal chemistry, 188, 10.1016/j.ejmech.2019.112005, 31911294
European journal of medicinal chemistry, 188, 10.1016/j.ejmech.2019.112005, 31911294
Novel PqsR Inverse Agonists
Publication
Hamed M,
Ahmed S,
Empting. M.,
Schütz C,
Hartmann R,
Röhrig T,
Kany A,
Hirsch A
(2020)
Patent, EP20150119/WO2021136805A1
Patent, EP20150119/WO2021136805A1
Toxic effect and genotoxicity of carvacrol ethers in Drosophila melanogaster
Publication
Nesterkina M,
Bilokon S,
Alieksieieva T,
Chebotar S,
Kravchenko I
(2020)
Mutat. Res., 821, 2, 10.1016/j.mrfmmm.2020.111713, 32593030
Mutat. Res., 821, 2, 10.1016/j.mrfmmm.2020.111713, 32593030