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Sorangicin A Is Active against Chlamydia in Cell Culture, Explanted Fallopian Tubes, and Topical In Vivo Treatment
Publication
Graspeuntner S,
Koethke K,
Scholz C,
Semmler L,
Lupatsii M,
Kirchhoff L,
Herrmann J,
Rox K,
Wittstein K,
Käding N,
Hanker L,
Stadler M,
Brönstrup M,
Müller R,
Shima K,
Rupp J
(2023)
Antibiotics, 12, 5, 10.3390/antibiotics12050795
Antibiotics, 12, 5, 10.3390/antibiotics12050795
In Vivo Activity Profiling of Biosynthetic Darobactin D22 against Critical Gram-Negative Pathogens
Publication
Kany A,
Fries F,
Seyfert C,
Porten C,
Deckarm S,
Chacón Ortiz M,
Dubarry N,
Vaddi S,
Große M,
Bernecker S,
Sandargo B,
Müller A,
Bacqué E,
Stadler M,
Herrmann J,
Müller R
(2024)
ACS Infect. Dis., 10, 12, 4337-4346, 10.1021/acsinfecdis.4c00687, 39565008
ACS Infect. Dis., 10, 12, 4337-4346, 10.1021/acsinfecdis.4c00687, 39565008
Regio- and Stereoselective Epoxidation and Acidic Epoxide Opening of Antibacterial and Antiplasmodial Chlorotonils Yield Highly Potent Derivatives
Publication
Müller R,
Hofer W,
Oueis E,
Abou Fayad A,
Deschner F,
Andreas A,
Carvalho L,
Hüttel S,
Bernecker S,
Pätzold L,
Morgenstern B,
Zaburannyi N,
Bischoff M,
Stadler M,
Held J,
Herrmann J
(2022)
Angewandte Chemie (International ed. in English), 10.1002/anie.202202816, 35485800
Angewandte Chemie (International ed. in English), 10.1002/anie.202202816, 35485800
Functionalization of Chlorotonils: Dehalogenil as Promising Lead Compound for In Vivo Application
Publication
Hofer W,
Deschner F,
Jézéquel G,
Pessanha de Carvalho L,
Abdel-Wadood N,
Pätzold L,
Bernecker S,
Morgenstern B,
Kany A,
Große M,
Stadler M,
Bischoff M,
Hirsch A,
Held J,
Herrmann J,
Müller R
(2024)
Angewandte Chemie (International ed. in English), 63, 19, 10.1002/anie.202319765, 38502093
Angewandte Chemie (International ed. in English), 63, 19, 10.1002/anie.202319765, 38502093
Pharmacology and early ADMET data of corallopyronin A, a natural product with macrofilaricidal anti-wolbachial activity in filarial nematodes
Publication
Ehrens A,
Schiefer A,
Krome A,
Becker T,
Rox K,
Neufeld H,
Aden T,
Wagner K,
Müller R,
Grosse M,
Stadler M,
König G,
Kehraus S,
Alt S,
Hesterkamp T,
Hübner M,
Pfarr K,
Hoerauf A
(2022)
Front. Trop. Dis, 3, 10.3389/fitd.2022.983107
Front. Trop. Dis, 3, 10.3389/fitd.2022.983107
Corallopyronin A: antimicrobial discovery to preclinical development
Publication
Krome A,
Becker T,
Kehraus S,
Schiefer A,
Gütschow M,
Chaverra-Muñoz L,
Hüttel S,
Jansen R,
Stadler M,
Ehrens A,
Pogorevc D,
Müller R,
Hübner M,
Hesterkamp T,
Pfarr K,
Hoerauf A,
Wagner K,
König G
(2022)
Nat. Prod. Rep., 10.1039/d2np00012a, 35730490
Nat. Prod. Rep., 10.1039/d2np00012a, 35730490
Amidochelocardin Overcomes Resistance Mechanisms Exerted on Tetracyclines and Natural Chelocardin
Publication
Hennessen F,
Miethke M,
Zaburannyi N,
Loose M,
Lukežic T,
Bernecker S,
Hüttel S,
Jansen R,
Schmiedel J,
Fritzenwanker M,
Imirzalioglu C,
Vogel J,
Westermann A,
Hesterkamp T,
Stadler M,
Wagenlehner F,
Petkovic H,
Herrmann J,
Müller R
(2020)
Antibiotics, 9, 9, 10.3390/antibiotics9090619, 32962088
Antibiotics, 9, 9, 10.3390/antibiotics9090619, 32962088
Corallopyronin A for short-course anti-wolbachial, macrofilaricidal treatment of filarial infections
Publication
Schiefer A,
Hübner M,
Krome A,
Lämmer C,
Ehrens A,
Aden T,
Koschel M,
Neufeld H,
Chaverra-Muñoz L,
Jansen R,
Kehraus S,
König G,
Pogorevc D,
Müller R,
Stadler M,
Hüttel S,
Hesterkamp T,
Wagner K,
Pfarr K,
Hoerauf A
(2020)
PLoS Negl. Trop. Dis., 14, 12, 10.1371/journal.pntd.0008930, 33284808
PLoS Negl. Trop. Dis., 14, 12, 10.1371/journal.pntd.0008930, 33284808
Towards the sustainable discovery and development of new antibiotics
Publication
Miethke M,
Pieroni M,
Weber T,
Brönstrup M,
Hammann P,
Halby L,
Arimondo P,
Glaser P,
Aigle B,
Bode H,
Moreira R,
Li Y,
Luzhetskyy A,
Medema M,
Pernodet J,
Stadler M,
Tormo J,
Genilloud O,
Truman A,
Weissman K,
Takano E,
Sabatini S,
Stegmann E,
Brötz-Oesterhelt H,
Wohlleben W,
Seemann M,
Empting M,
Hirsch A,
Loretz B,
Lehr C,
Titz A,
Herrmann J,
Jaeger T,
Alt S,
Hesterkamp T,
Winterhalter M,
Schiefer A,
Pfarr K,
Hoerauf A,
Graz H,
Graz M,
Lindvall M,
Ramurthy S,
Karlén A,
van Dongen M,
Petkovic H,
Keller A,
Peyrane F,
Donadio S,
Fraisse L,
Piddock L,
Gilbert I,
Moser H,
Müller R
(2021)
Nature reviews. Chemistry, 5, 10, 726-749, 10.1038/s41570-021-00313-1, 34426795
Nature reviews. Chemistry, 5, 10, 726-749, 10.1038/s41570-021-00313-1, 34426795