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The Structures and Binding Modes of Small-Molecule Inhibitors of Pseudomonas aeruginosa Elastase LasB
Publikation
Camberlein V,
Jézéquel G,
Haupenthal J,
Hirsch A
(2022)
Antibiotics, 11, 8, 10.3390/antibiotics11081060
Antibiotics, 11, 8, 10.3390/antibiotics11081060
Design, Synthesis, Antimicrobial Activity, and Molecular Docking of Some New Diclofenac Derivatives
Publikation
Tolba M,
Hamed M,
Sayed M,
Kamal El-Dean A,
Abdel-Mohsen S,
Ibrahim O,
Elgaher W,
Hirsch A,
Saddik A
(2022)
Polycyclic Aromatic Compounds, 1-16, 10.1080/10406638.2022.2102661
Polycyclic Aromatic Compounds, 1-16, 10.1080/10406638.2022.2102661
N-Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases
Publikation
Kaya C,
Konstantinovic J,
Kany A,
Andreas A,
Kramer J,
Brunst S,
Weizel L,
Rotter M,
Frank D,
Yahiaoui S,
Müller R,
Hartmann R,
Haupenthal J,
Proschak E,
Wichelhaus T,
Hirsch A
(2022)
Journal of medicinal chemistry, 65, 5, 3913-3922, 10.1021/acs.jmedchem.1c01755, 35188771
Journal of medicinal chemistry, 65, 5, 3913-3922, 10.1021/acs.jmedchem.1c01755, 35188771
Design and Synthesis of Novel Bis-Imidazolyl Phenyl Butadiyne Derivatives as HCV NS5A Inhibitors
Publikation
Hamdy J,
Emadeldin N,
Hamed M,
Frakolaki E,
Katsamakas S,
Vassilaki N,
Zoidis G,
Hirsch A,
Abdel-Halim M,
Abadi A
(2022)
Pharmaceuticals, 15, 5, 10.3390/ph15050632, 35631457
Pharmaceuticals, 15, 5, 10.3390/ph15050632, 35631457
N-Aryl-2-iso-butylmercaptoacetamides: the discovery of highly potent and selective inhibitors of Pseudomonas aeruginosa virulence factor LasB and Clostridium histolyticum virulence factor ColH
Publikation
Voos K,
Yahiaoui S,
Konstantinovic J,
Schönauer E,
Alhayek A,
Sikandar A,
Si Chaib K,
Ramspoth T,
Rox K,
Haupenthal J,
Köhnke J,
Brandstetter H,
Ducho C,
Hirsch A
(2022)
ChemRxiv, 10.26434/chemrxiv-2022-fjrqr
ChemRxiv, 10.26434/chemrxiv-2022-fjrqr
Inhibition of Collagenase Q1 of Bacillus cereus as a Novel Antivirulence Strategy for the Treatment of Skin‐Wound Infections
Publikation
Alhayek A,
Khan E,
Schönauer E,
Däinghaus T,
Shafiei R,
Voos K,
Han M,
Ducho C,
Posselt G,
Wessler S,
Brandstetter H,
Haupenthal J,
del Campo A,
Hirsch A
(2022)
Adv. Therap., 10.1002/adtp.202100222
Adv. Therap., 10.1002/adtp.202100222
Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor
Publikation
Drost M,
Diamanti E,
Fuhrmann K,
Goes A,
Shams A,
Haupenthal J,
Koch M,
Hirsch A,
Fuhrmann G
(2022)
Pharmaceutics, 14, 1, 10.3390/pharmaceutics14010004
Pharmaceutics, 14, 1, 10.3390/pharmaceutics14010004
Synthesis, biological evaluation, and molecular docking studies of aldotetronic acid-based LpxC inhibitors
Publikation
Wimmer S,
Hoff K,
Martin B,
Grewer M,
Denni L,
Lascorz Massanet R,
Raimondi M,
Bülbül E,
Melesina J,
Hotop S,
Haupenthal J,
Rohde H,
Heisig P,
Hirsch A,
Brönstrup M,
Sippl W,
Holl R
(2022)
Bioorganic chemistry, 131, 10.1016/j.bioorg.2022.106331, 36587505
Bioorganic chemistry, 131, 10.1016/j.bioorg.2022.106331, 36587505
New Ketene Dithioacetals Generated from 2-Nitroperchlorobutadiene and Investigation of Their Antibacterial, Antifungal, Anticonvulsant and Antidepressant Activities
Publikation
Aydinli S,
Bulut E,
Deniz N,
Sayil C,
Komarovska-Porokhnyavets O,
Lubenets V,
Zvarych V,
Stasevych M,
Nesterkina M,
Kravchenko I
(2022)
Chemistry & Biodiversity, 19, 7, 10.1002/cbdv.202100931, 35674435
Chemistry & Biodiversity, 19, 7, 10.1002/cbdv.202100931, 35674435
Discovery and Characterization of Synthesized and FDA-Approved Inhibitors of Clostridial and Bacillary Collagenases
Publikation
Alhayek A,
Abdelsamie A,
Schönauer E,
Camberlein V,
Hutterer E,
Posselt G,
Serwanja J,
Blöchl C,
Huber C,
Haupenthal J,
Brandstetter H,
Wessler S,
Hirsch A
(2022)
Journal of medicinal chemistry, 65, 19, 12933-12955, 10.1021/acs.jmedchem.2c00785, 36154055
Journal of medicinal chemistry, 65, 19, 12933-12955, 10.1021/acs.jmedchem.2c00785, 36154055