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Synthesis and Anticonvulsant Activity of New Calix[4]Arene Derivatives Containing Gamma-Aminobutyric Acid Moieties
Publikation
Nesterkina M,
Alekseeva E,
Kravchenko I
(2016)
Pharm Chem J, 49, 12, 825-829, 10.1007/s11094-016-1380-7
Pharm Chem J, 49, 12, 825-829, 10.1007/s11094-016-1380-7
Proteoid Dynamers with Tunable Properties
Publikation
Liu Y,
Stuart M,
Buhler E,
Lehn J,
Hirsch A
(2016)
, 10.1002/ADFM.201601612
, 10.1002/ADFM.201601612
Towards the evaluation in an animal disease model: Fluorinated 17β-HSD1 inhibitors showing strong activity towards both the human and the rat enzyme
Publikation
Abdelsamie A,
Bey E,
Gargano E,
van Koppen C,
Empting M,
Frotscher M
(2015)
European journal of medicinal chemistry, 103, 56-68, 10.1016/j.ejmech.2015.08.030, 26322835
European journal of medicinal chemistry, 103, 56-68, 10.1016/j.ejmech.2015.08.030, 26322835
Novel PqsR Inverse Agonists
Publikation
Hamed M
(2015)
Patent, EP 201523196
Patent, EP 201523196
Fragment growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin
Publikation
Mondal M,
Groothuis D,
Hirsch A
(2015)
, 10.1039/C5MD00157A
, 10.1039/C5MD00157A
Validation of a homology model of Mycobacterium tuberculosis DXS: rationalization of observed activities of thiamine derivatives as potent inhibitors of two orthologues of DXS
Publikation
Masini T,
Lacy B,
Monjas L,
Hawksley D,
Voogd A,
Illarionov B,
Iqbal A,
Leeper F,
Fischer M,
Kontoyianni M,
Hirsch A
(2015)
Organic & biomolecular chemistry, 13, 46, 11263-77, 10.1039/c5ob01666e, 26411373
Organic & biomolecular chemistry, 13, 46, 11263-77, 10.1039/c5ob01666e, 26411373
Structure-based design of potent small-molecule binders to the S-component of the ECF transporter for thiamine
Publikation
Swier L,
Monjas L,
Guskov A,
Voogd A,
Erkens G,
slotboom d,
Hirsch A
(2015)
ChemBioChem, 16, 5, 819-26, 10.1002/cbic.201402673, 25676607
ChemBioChem, 16, 5, 819-26, 10.1002/cbic.201402673, 25676607
Fighting malaria: structure-guided discovery of nonpeptidomimetic plasmepsin inhibitors
Publikation
Huizing A,
Mondal M,
Hirsch A
(2015)
Journal of medicinal chemistry, 58, 13, 5151-63, 10.1021/jm5014133, 25719272
Journal of medicinal chemistry, 58, 13, 5151-63, 10.1021/jm5014133, 25719272
Supramolecular chemistry … and beyond
Publikation
Hirsch A
(2015)
Angewandte Chemie (International ed. in English), 54, 38, 11013-4, 10.1002/anie.201506536, 26306880
Angewandte Chemie (International ed. in English), 54, 38, 11013-4, 10.1002/anie.201506536, 26306880
Engineering a Constrained Peptidic Scaffold towards Potent and Selective Furin Inhibitors
Publikation
Fittler H,
Depp A,
Avrutina O,
Dahms S,
Than M,
Empting M,
Kolmar H
(2015)
Chembiochem : a European journal of chemical biology, 16, 17, 2441-4, 10.1002/cbic.201500447, 26426719
Chembiochem : a European journal of chemical biology, 16, 17, 2441-4, 10.1002/cbic.201500447, 26426719