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Design and Synthesis of Bioisosteres of Acylhydrazones as Stable Inhibitors of the Aspartic Protease Endothiapepsin
Publikation
Jumde V,
Mondal M,
Gierse R,
Unver M,
Magari F,
van Lier R,
Heine A,
Klebe G,
Hirsch A
(2018)
ChemMedChem, 13, 21, 2266-2270, 10.1002/cmdc.201800446
ChemMedChem, 13, 21, 2266-2270, 10.1002/cmdc.201800446
Delivery system for budesonide based on lipid-DNA
Publikation
Liu Y,
Bos I,
Oenema T,
Meurs H,
Maarsingh H,
Hirsch A
(2018)
European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 130, 123-127, 10.1016/j.ejpb.2018.06.012, 29908939
European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 130, 123-127, 10.1016/j.ejpb.2018.06.012, 29908939
Dynamic Proteoids Generated From Dipeptide-Based Monomers
Publikation
Liu Y,
Stuart M,
Buhler E,
Hirsch A
(2018)
Macromolecular rapid communications, 39, 13, 10.1002/marc.201800099, 29806088
Macromolecular rapid communications, 39, 13, 10.1002/marc.201800099, 29806088
Phage Display on the Anti-infective Target 1-Deoxy-d-xylulose-5-phosphate Synthase Leads to an Acceptor-Substrate Competitive Peptidic Inhibitor
Publikation
Marcozzi A,
Masini T,
Di Zhu,
Pesce D,
Illarionov B,
Fischer M,
Herrmann A,
Hirsch A
(2018)
ChemBioChem, 19, 1, 58-65, 10.1002/cbic.201700402, 29119720
ChemBioChem, 19, 1, 58-65, 10.1002/cbic.201700402, 29119720
Generation of Semi-Synthetic Shark IgNAR Single-Domain Antibody Libraries
Publikation
Grzeschik J,
Könning D,
Hinz S,
Krah S,
Schröter C,
Empting M,
Kolmar H,
Zielonka S
(2018)
Methods in molecular biology (Clifton, N.J.), 1701, 147-167, 10.1007/978-1-4939-7447-4_8, 29116504
Methods in molecular biology (Clifton, N.J.), 1701, 147-167, 10.1007/978-1-4939-7447-4_8, 29116504
Donepezil-melatonin hybrids as butyrylcholinesterase inhibitors: Improving binding affinity through varying mode of linking fragments
Publikation
Lozinska I,
Swierczynska A,
Moleda Z,
Hartman A,
Hirsch A,
Czarnocki Z
(2018)
Archiv der Pharmazie, 351, 11, 10.1002/ardp.201800194, 30290008
Archiv der Pharmazie, 351, 11, 10.1002/ardp.201800194, 30290008
Repellent activity of monoterpenoid esters with neurotransmitter amino acids against yellow fever mosquito, Aedes aegypti
Publikation
Nesterkina M,
Bernier U,
Tabanca N,
Kravchenko I
(2018)
Open Chemistry, 16, 1, 95-98, 10.1515/chem-2018-0015
Open Chemistry, 16, 1, 95-98, 10.1515/chem-2018-0015
Trendbericht Biochemie 2017: Proteinvermittelte dynamische kombinatorische Chemie
Publikation
Hirsch A
(2018)
Nachr. Chem., 66, 3, 281-283, 10.1002/nadc.20184071734
Nachr. Chem., 66, 3, 281-283, 10.1002/nadc.20184071734
Insight into the complete substrate-binding pocket of ThiT by chemical and genetic mutations
Publikation
Swier L,
Monjas L,
Reeßing F,
Oudshoorn R,
Aisyah,
Primke T,
Bakker M,
van Olst E,
Ritschel T,
Faustino I,
Marrink S,
Hirsch A,
Slotboom D
(2017)
MedChemComm, 8, 5, 1121-1130, 10.1039/c7md00079k, 30108823
MedChemComm, 8, 5, 1121-1130, 10.1039/c7md00079k, 30108823
Saccharide-Containing Dynamic Proteoids
Publikation
Liu Y,
Stuart M,
Witte M,
Buhler E,
Hirsch A
(2017)
Chemistry (Weinheim an der Bergstrasse, Germany), 23, 64, 16162-16166, 10.1002/chem.201703584, 28981987
Chemistry (Weinheim an der Bergstrasse, Germany), 23, 64, 16162-16166, 10.1002/chem.201703584, 28981987